SLC22A8 (Organic anion transporter 3) variants and mutations

SLC22A8 (also known as Organic anion transporter 3) is a human protein-coding gene encoding an organic anion transporter 3 protein. It transports a broad range of organic anions from blood into renal proximal-tubule cells for secretion into urine. It is an important determinant of renal clearance and drug-drug interactions for numerous medications and endogenous metabolites. This analysis covers 956 SLC22A8 variants and mutations. Of these, 90% have computational variant effect predictions. Disease context includes gout, Hypertension, and endothelial dysfunction. Example SLC22A8 variants include M1?, S4*, and S4L.

Variant analysis overview

Variant and mutation evidence

Clinical, disease, and population context

Protein structure and variant hotspots

Data sources

Evidence in this analysis draws on EBI Proteins Variation, UniProt, gnomAD v4, EuropePMC, 3D Hotspot Analysis, Interaction Network Analysis, AlphaFold DB, gnomAD constraint, Open Targets, MaveDB, LitVar.

Notable SLC22A8 variants

Examples include M1?, S4*, S4L, E5G, E5K, D8H, D8N, R9C. Listed records include available protein-change notation, database identifiers, clinical classifications, computational predictions, population evidence, experimental measurements, and disease context.